Yayıncı "Elsevier France-Editions Scientifiques Medicales Elsevier" için listeleme
Toplam kayıt 46, listelenen: 1-20
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0-1 integer programming model for procedural separation of aircraft by ground holding in ATFM
(Elsevier France-Editions Scientifiques Medicales Elsevier, 2014)This study presents a 0-1 integer programming model for air traffic flow management. The model is used for determining optimum departure times of aircraft so as to avoid aircraft conflicts and to balance capacity and demand ... -
Anticandidal pimaradiene diterpene from Phlomis essential oils
(Elsevier France-Editions Scientifiques Medicales Elsevier, 2009)In the present study, it was aimed to investigate the phytochemical profile and antimicrobial effects of Phlomis lunariifolia Sm., Phlomis amanica Vierh., Phlomis monocephala P.H. Davis, Phlomis sieheana Rech. fil, Phlomis ... -
Antimicrobial activity and a SAR study of some novel benzimidazole derivatives bearing hydrazone moiety
(Elsevier France-Editions Scientifiques Medicales Elsevier, 2010)In this study 12 novel benzimidazole compounds bearing hydrazone moiety were synthesized in order to investigate their possible antibacterial and antifungal activity. Structures of the synthesized compounds were elucidated ... -
A comparison of the ground reaction forces of archers with different levels of expertise during the arrow shooting
(Elsevier France-Editions Scientifiques Medicales Elsevier, 2019)Objective. - The purpose of this study was to compare the differences in ground reaction forces (GRFs) of archers with different levels of expertise during arrow shooting. Material and methods. - Twenty-seven male archers ... -
Cytotoxic and genotoxic effects of [Ru(phi)(3)](2+) evaluated by Ames/Salmonella and MTT methods
(Elsevier France-Editions Scientifiques Medicales Elsevier, 2009)In this work, we synthesized and evaluated the cytotoxic effect of [Ru(phi)(3)](2+), on rat C6 glioma cell line. Cell viability was determined by assay with 3-(4-5-dimethylthiazol-2-yl)-2,5-diphenyl tetrazolium bromide ... -
Design, synthesis and biological assessment of new thiazolylhydrazine derivatives as selective and reversible hMAO-A inhibitors
(Elsevier France-Editions Scientifiques Medicales Elsevier, 2018)In the recent works, it was shown that numerous thiazolylhydrazine derivatives display hMAO inhibitory activity in the range of micromolar concentration. Hence, in the present study a new series of new thiazole-hydrazines ... -
Design, synthesis, in vitro and in silico evaluation of a new series of oxadiazole-based anticancer agents as potential Akt and FAK inhibitors
(Elsevier France-Editions Scientifiques Medicales Elsevier, 2018)In the current work, new 1,3,4-oxadiazole derivatives were synthesized and investigated for their cytotoxic effects on A549 human lung adenocarcinoma, C6 rat glioma and NIH/3T3 mouse embryonic fibroblast cell lines. Compounds ... -
DFT, FT-Raman, FT-IR, solution and solid state NMR studies of 2,4-dimethoxyphenylboronic acid
(Elsevier France-Editions Scientifiques Medicales Elsevier, 2011)The possible stable forms and molecular structures of 2,4-dimethoxyphenylboronic acid (2,4-dmpba) have been experimentally and theoretically studied using FT-IR. Raman and solution and solid state NMR spectroscopic methods. ... -
Fuel flow analysis for the cruise phase of commercial aircraft on domestic routes
(Elsevier France-Editions Scientifiques Medicales Elsevier, 2014)From the point of view of the environmental impact of aviation, rather than fundamental strategies mainly intended for lower fuel consumption, and thereby less carbon dioxide emissions, more comprehensive approaches have ... -
Indomethacin based new triazolothiadiazine derivatives: Synthesis, evaluation of their anticancer effects on T98 human glioma cell line related to COX-2 inhibition and docking studies
(Elsevier France-Editions Scientifiques Medicales Elsevier, 2016)In the current work, new 1,2,4-triazolo[3,4-b]-1,3,4-thiadiazine derivatives (1-8) were synthesized via the ring closure reaction of 2-bromoacetophenone derivatives with 4-amino-5-[(5-methoxy-2-methyl-1(4-chlorobenzoyl)- ... -
MAO enzymes inhibitory activity of new benzimidazole derivatives including hydrazone and propargyl side chains
(Elsevier France-Editions Scientifiques Medicales Elsevier, 2017)In the present work, 15 new N'-(arylidene)-4-(1-(prop-2-yn-1-yl)-1H-benzo[dlimidazol-2-yl)benzohydrazide (4a-4o) were designed and synthesized. The structures of the synthesized compounds were elucidated using FT-IR, ... -
Microwave supported synthesis of some novel 1,3-Diarylpyrazino[1,2-a] benzimidazole derivatives and investigation of their anticancer activities
(Elsevier France-Editions Scientifiques Medicales Elsevier, 2011)The syntheses of 1,3-diarylpyrazino[1,2-a]benzimidazole derivatives and the investigation of their anticancer activities were studied. For this, 2-aryloylbenzimidazole derivatives were reacted with 2-bromoacetophenones in ... -
Modeling the fuel flow-rate of transport aircraft during flight phases using genetic algorithm-optimized neural networks
(Elsevier France-Editions Scientifiques Medicales Elsevier, 2016)Predicting the fuel consumption of transport aircraft is vital for minimizing the detrimental effects of fuel emissions on the environment, saving fuel energy sources, reducing flight costs, achieving more accurate aircraft ... -
Molecular structure, NMR analyses, density functional theory and ab initio Hartree-Fock calculations of 3-phenylpropylamine
(Elsevier France-Editions Scientifiques Medicales Elsevier, 2009)H-1, C-13, DEPT, COSY, NOESY and HETCOR NMR spectra of 3-phenylpropylamine (3-PPA) have been reported in chloroform-d, dichloromethane-d, methanol-d, dimethylsulfoxide-d and acetone-d. Solvent effects on nuclear magnetic ... -
New piperidine-hydrazone derivatives: Synthesis, biological evaluations and molecular docking studies as AChE and BChE inhibitors
(Elsevier France-Editions Scientifiques Medicales Elsevier, 2016)Hydrazones and the piperidine ring containing compounds were considered as beneficial substrates in drug design. Therefore, this study was aimed at the synthesis of new benzoyl hydrazones derived from ethyl 4-oxopiperidi ... -
New pyrazoline derivatives and their antidepressant activity
(Elsevier France-Editions Scientifiques Medicales Elsevier, 2010)Some triazolo-pyrazoline derivatives were synthesized to investigate their potential antidepressant activities. The chemical structures of the compounds were elucidated by IR, NMR and FAB(+)-MS spectral data and elemental ... -
New triazole and triazolothiadiazine derivatives as possible antimicrobial agents
(Elsevier France-Editions Scientifiques Medicales Elsevier, 2008)Triazole and triazoles fused with six-membered ring systems are found to possess diverse applications in the fields of medicine, agriculture and industry. The new 1,2,4-triazole and 1,2,4-triazolo[3,4-b][1,3,4]thiadiazine ... -
A novel series of thiazolyl-pyrazoline derivatives: Synthesis and evaluation of antifungal activity, cytotoxicity and genotoxicity
(Elsevier France-Editions Scientifiques Medicales Elsevier, 2015)In the current work, new thiazolyl pyrazoline derivatives (1-22) were synthesized and evaluated for their antifungal effects against pathogenic yeasts and molds using a broth microdilution assay. Ames assay was carried out ... -
Numerical optimization of a fin-tube gas to liquid heat exchanger
(Elsevier France-Editions Scientifiques Medicales Elsevier, 2012)The influence of plate fin, fin tube and protrusion parameters on heat transfer and pressure drop characteristics of a finned tube gas to liquid heat exchanger is examined in this study. The optimization of plate fin, fin ... -
Oxidative stress and mRNA expression of acetylcholinesterase in the leukocytes of ischemic patients
(Elsevier France-Editions Scientifiques Medicales Elsevier, 2017)Background: Pathogenesis of ischemic brain injury is occurred by crucial metabolic reasons. For instance, oxidative stress from free radical generation is causing to the thrombotic cerebrovascular stroke. In this case, the ...