Thioamidoalkylation of 1,3-dicarbonyl compounds, enol silyl ethers, and enamines

Abstract

Novel syntheses of beta-thioamido ketones via thioamidoalkylations of malonates, beta-keto esters, beta-diketones, enol silyl ethers, and enamines with N-(alpha-thioamidoalkyl)benzotriazoles are described.