Başlık için Eczacılık Fakültesi listeleme
Toplam kayıt 1731, listelenen: 1334-1353
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Simultaneous Determination of Substance P and CGRP in Rat Brainstem Tissue Using LC-ESI-MS/MS Method
(Bentham Science Publ LTD, 2018)Background: Substance P and CGRP are neuropeptides that belong to the thachykinin and calcitonin family, respectively. They play an important role in neuropathic pain development and regulation. Methods: In this study, ... -
Sitophilus granarius L. (Coleoptera) Toxicity and Biological Activities of the Essential Oils of Tanacetum macrophyllum (Waldst. & Kit.) Schultz Bip.
(Japan Oil Chemists Soc, 2015)Insecticides of the natural origin are an important alternative to the synthetic insecticides that are being employed for the preserving stored products. The volatiles obtained from T. cinerariifolium (=Pyrethrum ... -
Solid lipid and chitosan particulate systems for delivery of siRNA
(Govi-Verlag Pharmazeutischer Verlag GMBH, 2015)Due to the recent advances in molecular biology, there are promising gene therapy studies for prevention and treatment of cancer, genetic and infectious diseases. Many technologies in molecular biology and biotechnology ... -
Solid lipid nanoparticles: A possible vehicle for zinc oxide and octocrylene
(Govi-Verlag Pharmazeutischer Verlag GMBH, 2012)An efficient sunscreen formulation shows good absorption in the relevant UV range. Efficacy also means that the UV absorber must be easily incorporated in any kind of formulation. In this study, a chemical absorber, ... -
Solid lipid non-particles (SLN) [Kati lipit nanopartiküller (SLN)]
(2000)Colloidal drug delivery systems are one of the subjects investigated intensively in the pharmaceutical field, in recent years. Those systems include microspheres, polymeric nanoparticles, liposomes and fat emulsions. An ... -
Some 1-substituted 3-aryl-1,4-dihydro-1,2,4-triazino[4,3-a]- benzimidazoles and their vasodilatory activities
(Societa Chimica Italiana, 1997)In this study, some 1-substituted 3-aryl-1,4-dihydro-1,2,4- triazino[4,3-a]benzimidazole derivatives were synthesized, their structures were elucidated, and their vasodilatory activities were examined. It was found that ... -
Some 3-alkyl-6-(2-aryl-2-oxo-1-ethyl)-7-oxothiazolo [4,5-d]pyrimidin-2(3H)-thione derivatives and their antimicrobial activities
(2005)In this study, some 3-alkyl-6-(2-aryl-2-oxo-1-ethyl)-7-oxothiazolo [4,5-d]pyrimidin-2(3H)-thione derivatives have been synthesized by reacting 3-alkyl-7-oxothiazolo[4,5-d]pyrimidin-2(3H)-thiones with various ?-bromoacetophenones. ... -
Some 6-substituted 3-aryl-7-oxothiazolo[4,5-d]pyrimidin-2(3H)-thione derivatives and their antimicrobial activities
(Taylor & Francis LTD, 2007)In this study, 3-aryl-6-substituted thiazolopyrimidin-2(3H)-thione derivatives 4 and 6 have been synthesized by reacting thiazolopyrimidines 2 with omega-bromoacetophenone 3 and 2-chloro-N-(2-thiazolyl)acetamides 5. The ... -
Some new 2,3-dihydro-3 benzofuranamine derivatives
(1998)In this study, four series of the compounds (i.e. 2, 3, 4 and 5) were synthesized using the 2-chloro-N-(2,3-dihydro-3-benzofuryl)acetamides. The structures of the compounds were elucidated by IR, 1H-NMR, MASS spectroscopy ... -
Some new 4-aryl-2-thiazolylhydrazones
(1997)In this study, three series of 4-aryl-2-thiazolylhydrazones were synthesized using three different thiosemicarbazones. Structures of the compounds were elucidated by IR, 1H NMR and elemental analysis. The prepared compounds ... -
Some new 7-aryloxyalkyltheophyllines as bronchodilators
(Editions Scientifiques Medicales Elsevier, 1997)… -
Some nitroimidazole derivatives as possible antibacterial agents
(1993)In this study, six 1-[2(benzazol-2-yl)thioethy-2-methyl-5-nitroimidazole derivatives were synthesized. Antibacterial activities of the compounds obtained were examined and it was found that they are effective against aerobe ... -
Some phytochemical investigations of jerusalem sage (Phlomis pungens Willd.) [TİKANLI ODOTU (Phlomis pungens Willd.) NÖVÜNÜN Binverted eZİ FİTOKİMYinverted eVİ Tinverted eDQİQİ]
(Azerbaijan Medical University, 2013)The results of phytochemical investigation of Jerusalem Sage distributed in Azerbaijan obtained the present of the phenolic compounds sum and essential oils. The 3 individual substances were isolated from the phenolic ... -
Some pyridazinone and phthalazinone derivatives and their vasodilator activities
(Pharmaceutical Society of Korea, 2004)In this study, 6-[(4-arylidene-2-phenyl-5-oxoimidazolin-1-yl)phenyl]-4,5- dihydro-3(2H)-pyridazinone and 4-[(4-arylidene-2-phenyl-5-oxoimidazolin-1-yl) phenyl]-1(2H)-phthalazinone derivatives were synthesized by reacting ... -
Some pyrrole substituted aryl pyridazinone and phthalazinone derivatives and their antihypertensive activities
(2004)In this work, some 2-nonsubstituted/2-methyl-/2-(2-acetyloxyethyl)-6-[4- (substituted pyrrol-1-yl)phenyl]-4,5-dihydro-3(2H)-pyridazinone, derivatives and 2-nonsubstituted/2-methyl- 4-[4-(substituted pyrrol-1-yl)phenyl]-1(2H)- ... -
Some Thiazole Derivatives Combined with Different Heterocycles: Cytotoxicity Evaluation and Apoptosis Inducing Studies
(Bentham Science Publ LTD, 2018)Background: Thiazole ring is an outstanding structure found in many biologically active compounds and clinically available drugs. Because of synthesis simplicity of its derivatives and having a wide range of biological ... -
Some thiazolylaminopyrrole derivatives and their antimicrobial activity
(1999)In this study, some ethyl 1-(4-arylthiazol-2-yl)amino-2-methyl-5-aryl-1H-pyrrole-3-carboxylic acid derivatives were obtained by reacting 1-(2-methyl-3-carbethoxy-5-arylpyrrol-1-yl)thioureas with ?-bromoacetophenone ... -
Spectral, electrochemical and DFT studies of a trimetallic Cu-II Derivative: Antimycobacterial and cytotoxic activity
(Elsevier Science Sa, 2019)The trimetallic Cu-II derivative, [Cu-3(L)(2)(ClO4)(2)] (1) [where H2L = N,N'-bis(salicylidene)-1,3-propanediamine] has been synthesized and characterized by different spectral techniques. In 1, the two terminal Cu-II atoms ... -
Spectroscopic Determination and Evaluation of Acidity Constants for Some Drug Precursor 2-Amino-4-(3-or 4-substituted phenyl) Thiazole Derivatives
(American Chemical Society, 2010)Acid dissociation constants, K(a), of eight drug precursor 2-amino-4-(3- or 4-substituted phenyl) thiazole derivatives were determined using a UV-vis spectroscopic technique. The obtained K(a) values were evaluated by ... -
Spectroscopic determination of acid dissociation constants of some biologically active 6-phenyl-4,5-dihydro-3(2H)-pyridazinone derivatives
(American Chemical Society, 2002)The acid dissociation constants, pK(a), of twelve biologically active 6-phenyl-4,5-dihydro-3(2H)-pyridazinone derivatives were determined using spectroscopic techniques. Elucidation of the structure-reactivity relationships ...