Güncel Gönderiler: Eczacılık Fakültesi
Toplam kayıt 1731, listelenen: 501-520
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Synthesis and biological evaluation of new naphthalene substituted thiosemicarbazone derivatives as potent antifungal and anticancer agents
(Elsevier France-Editions Scientifiques Medicales Elsevier, 2016)New thiosemicarbazone derivatives (1-10) were obtained via the reaction of 4-(naphthalen-1-yl)thiosemicarbazide with fluoro-substituted aromatic aldehydes. The synthesized compounds were evaluated for their in vitro ... -
Synthesis and Mosquitocidal Activity of a Series of Hydrazone Derivatives against Aedes aegypti
(Bentham Science Publ LTD, 2018)Background: Aedes aegypti is an important mosquito vector for the transmission of several infectious diseases. Current insecticides play a vital role in controlling mosquitoes; however, the frequent use of insecticides has ... -
Synthesis and anticandidal activity of new triazolothiadiazine derivatives
(Elsevier France-Editions Scientifiques Medicales Elsevier, 2011)New triazolothiadiazine derivatives were synthesized via the ring closure reaction of 4-amino-5-substituted-2,4-dihydro-3H-1,2,4-triazol-3-thiones with phenacyl bromides. The compounds were tested in vitro against various ... -
Synthesis and Anticholinesterase Activity and Cytotoxicity of Novel Amide Derivatives
(Wiley-V C H Verlag GMBH, 2012)In the present study, some amide derivatives were synthesized and their potential anticholinesterase properties were investigated. N-(Benzothiazol-2-yl)-2-[(5-amino/methyl-1,3,4-thiadiazol-2-yl)thio]acetamide derivatives ... -
Synthesis of Some Novel Triazole Derivatives and Investigation of Their Antimicrobial Activities
(Taylor & Francis Inc, 2011)[image omitted] The aim of this study is to synthesize new triazole derivatives and investigate their antimicrobial activities. 4-Amino-5-(2-cyclohexylethyl)-3-[N-(benzothiazole-2-yl)acetamido]thio-4H-1,2,4-triazole and ... -
Synthesis and Evaluation of New 1,3,4-Thiadiazole Derivatives as Antinociceptive Agents
(MDPI AG, 2016)In the current work, new 1,3,4-thiadiazole derivatives were synthesized and investigated for their antinociceptive effects on nociceptive pathways of nervous system. The effects of these compounds against mechanical, thermal ... -
Synthesis and Evaluation of a Series of 1,3,4-Thiadiazole Derivatives as Potential Anticancer Agents
(Bentham Science Publ LTD, 2018)Background and Methods: In an attempt to develop potent antitumor agents, the synthesis of a series of N-(6-substituted benzothiazol-2-yl)-2-1(5-(arylamino)-1,3,4-thiadiazol-2-yl)thiolacetamides (1-14) was described and ... -
Synthesis and Biological Evaluation of a Series of Dithiocarbamates as New Cholinesterase Inhibitors
(Wiley-V C H Verlag GMBH, 2013)In the present paper, a novel series of dithiocarbamates was synthesized via the treatment of 4-(trifluoromethyl)benzyl chloride with appropriate sodium salts of N,N-disubstituted dithiocarbamic acids. H-1 NMR, mass spectral ... -
Novel imidazole derivatives as antifungal agents: Synthesis, biological evaluation, ADME prediction and molecular docking studies
(Taylor & Francis LTD, 2019)A series of 2-(substituteddithiocarbamoyl)-N-[4-((1H-imidazol-1-yl)methyl)phenyl]acetamide derivatives was designed and synthesized to combat the increasing incidence of drug-resistant fungal infections. All synthesized ... -
Design, synthesis, in vitro and in silico evaluation of new pyrrole derivatives as monoamine oxidase inhibitors
(Wiley-V C H Verlag GMBH, 2018)In an effort to develop potent monoamine oxidase (MAO) inhibitors, new pyrrole derivatives were obtained via the selective reduction of the CC bonds of 1-(1-methyl-1H-pyrrol-2-yl)-3-[5-(aryl)furan-2-yl]prop-2-en-1-ones ... -
Synthesis and Biological Evaluation of Some Pyrazoline Derivatives Bearing a Dithiocarbamate Moiety as New Cholinesterase Inhibitors
(Wiley-V C H Verlag GMBH, 2013)In the present study, new pyrazoline derivatives were synthesized via the reaction of 1-(chloroacetyl)-3-(2-furyl)-5-aryl-2-pyrazolines with sodium salts of N,N-disubstituted dithiocarbamic acids. Each derivative was ... -
Türkiye Aristolochia L. türlerinin yaprak morfolojisi ve anatomileri üzerinde çalışmalar
(1998)Türkiye Aristolochia türlerinin yaprak morfoloji ve anatomileri incelenmiştir. Anatomik çalışmalar yaprak laminası üzerinde yapılmıştır. Yaprak laminasının orta kısmından enine, üst ve alt yüzünden alınan yüzeysel kesitler ... -
Oltu (Erzurum) yöresinde halk ilacı olarak kullanılan tıbbi bitkiler
(2015)Bu çalışma Erzurum ili, Oltu ve yöresinde geleneksel halk ilacı olarak kullanılan bitkileri ortaya çıkarmak amacıyla yapılmıştır. Bu amaçla 2012 yılı temmuz ve ağustos aylarında, 2013 yılı şubat ve nisan aylarında arazi ... -
Seed morphology of some Genista taxa growing in Turkey
(2013)Birçok Angiosperm familyasında tohum makro ve mikromorfolojisi taksonomik öneme sahiptir. Bu çalışmada, Türkiye’de yetişen bazı Genista tohumlarının stero ve taramalı elekton mikroskobu (SEM) kullanılarak morfolojileri ... -
Öncesinde Acinos olarak bilinen Türkiye'deki altı Clinopodium taksonunun nutlet morfolojisi
(2014)Lamiaceae'nin Satureja, Calamintha, Micromeria, Clinopodium ve Acinos cinslerine ait türlerin bir grubu genel sınırları içinde karışıklığa neden olmaktadır. Bu çalışmada, öncesinde Acinos olarak bilinen Türkiye Florası'ndaki ... -
Taxonomical and morphological studies on the genus Calamintha Miller (Lamiaceae) in Turkey
(2009)Türkiye Florası’nda Calamintha Miller (Lamiaceae) cinsi 6’sı endemik olmak üzere 9 tür ve 13 takson ile temsil edilmektedir. Bu çalışmada Calamintha cinsine ait 13 takson sistematik ve morfolojik yönden incelenmiş, ... -
Nutlet surface micromorphology of the genus nepeta L.(lamiaceae) in Turkey
(2008)Nepeta L. cinsinin nutlet karakterleri taksonomik öneme sahiptir. Bu çalışmada, Türkiye'de yayılışı olan Nepeta türlerinin nutlet morfolojisi stereoskopik ve taramalı electron mikroskobu kullanılarak (SEM) incelenmiştir. ... -
Light effects on seed germination of endemic Centaurea L. species in section Phalolepıs (Cass.) DC
(2015)Dünya'da 600 Centaurea L. türü yayılış gösterirken, Avrupa'da 221 tür bulunmaktadır. Türkiye'de Astragalus L. ve Verbascum L. cinslerinden sonra Centaurea en çok türe sahip üçüncü cinstir. Endemizm oranı yüksektir ... -
Investigation of morphological, morphometric and anatomical characteristics of endemic Verbascum orgyale Boiss. & Heldr.
(2015)Anadolu'da "Sığır kuyruğu" olarak adlandırılan Verbascum L.(Scrophulariaceae) cinsi, ülkemizde 194'ü endemik olmak üzere 245 tür ile temsil edilmektedir. Çiçekleri müsilaj, uçucu yağ veglikozitlertaşır. Bazı Verbascum ...