Yazar "Durgun, Mustafa" için listeleme
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Benzenesulfonamide derivatives containing imine and amine groups: Inhibition on human paraoxonase and molecular docking studies
Isik, Mesut; Beydemir, Sukru; Demir, Yeliz; Durgun, Mustafa; Turkes, Cuneyt; Nasir, Abdul; Akkus, Musa (Elsevier, 2020)Sulfonamides known as inhibitors of many metabolic enzymes have been widely used as antimicrobial drugs for a long time. in the present study, we investigated in vitro inhibitory activities of benzenesulfonamide derivatives ... -
Molecular docking and investigation of 4-(benzylideneamino)- and 4-(benzylamino)-benzenesulfonamide derivatives as potent AChE inhibitors
Isik, Mesut; Demir, Yeliz; Durgun, Mustafa; Turkes, Cuneyt; Necip, Adem; Beydemir, Sukru (Springer International Publishing Ag, 2020)The discovery of acetylcholinesterase inhibitors is important for the treatment of Alzheimer's disease (AD), known as the most common type of dementia. Due to the side effects of commonly used acetylcholinesterase inhibitors, ... -
Synthesis, characterisation, biological evaluation and in silico studies of sulphonamide Schiff bases
Durgun, Mustafa; Turkes, Cuneyt; Isik, Mesut; Demir, Yeliz; Sakli, Ali; Kuru, Ali; Supuran, Claudiu T. (Taylor & Francis Ltd, 2020)Sulphonamides are biologically important compounds with low toxicity, many bioactivities and cost-effectiveness. Eight sulphonamide derivatives were synthesised and characterised by FT-IR, C-13 NMR, H-1 NMR, LC-MS and ... -
Synthesis, characterization, inhibition effects, and molecular docking studies as acetylcholinesterase, ?-glycosidase, and carbonic anhydrase inhibitors of novel benzenesulfonamides incorporating 1,3,5-triazine structural motifs
Lolak, Nebih; Akocak, Suleyman; Turkes, Cuneyt; Taslimi, Parham; Isik, Mesut; Beydemir, Sukru; Durgun, Mustafa (Academic Press Inc Elsevier Science, 2020)…
