Yazar "Erol, K" için listeleme
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1-N-substituted thiocarbamoyl-3-phenyl-5-thienyl-2-pyrazolines: Synthesis and evaluation as MAO inhibitors
Gökhan, N; Yeşilada, A; Uçar, G; Erol, K; Bilgin, AA (Wiley-V C H Verlag GMBH, 2003)Twelve new 1-N-substituted thiocarbomoyl-3-phehyl-5-thienyl-2-pyrazoline derivatives were synthesized and evaluated their for antidepressant, anxiogenic and mammalian monoamine oxidase (MAO)-A and B inhibitory activities ... -
3-Acetyl-4-Aryl-5-Oxo-2,7,7-Trimethyl-1,4,5,6,7,8-Hexahydroquinoline Derivatives and Their Calcium Antagonistic Activities
Şafak, C; ÖZKANLI, F; Erol, K; AKTAN, Y (Ecv-Editio Cantor Verlag Medizin Naturwissenschaften, 1995)Thirteen 3-acetyl-4-aryl-5-oxo-2,7,7-trimethyl-1,4,5,6,7,8-hexahydroquinoline derivatives (5a-m), one of which was synthesized before have been prepared. The structures of the products 5b-m were characterized by IR, H-1-NMR ... -
3-Aroylmethyl-2H-1,3-Benzoxazinedione Derivatives With Anticholinergic and Antihistaminic Activities
PilliayyIldız, Hg; Özkanli, F; Palaska, E; Şafak, C; Erdoğan, H; Erol, K; Özdemir, M (Soc Chimica Italiana, 1993)The synthesis of new 3-aroylmethyl-2H-1,3-benzoxazinedione derivatives is reported. The structure of these products are supported by their UV, IR and H-1-NMR spectra, as well as by elemental analysis. The new compounds ... -
5-methyl-8-N-substituted-thiocarbamoyl-7,8-diazabicyclo[4.3.0] non-6-enes: Evaluation as BSAO inhibitors and pharmacological activity screening
Yeşilada, A; Gökhan, N; Özer, I; Vural, K; Erol, K (Soc Chimica Italiana, 1996)In this study a series of 5-methyl-8-N-substituted-thiocarbamoyl-7,8-diazabicyclo[4.3.0] non-6-enes derivatives previously synthesized and separated to their stereoisomers, were evaluated as BSAO inhibitors and screened ... -
Analgesic and Anti-Inflammatory Effects of Some Benzanilides
Oskay, E; Aksu, F; Cingi, Mi; Erol, K; Fidan, Mehmet (Amer Pharmaceutical Assn, 1989)… -
Effects of Capsaicin on Isolated Guinea-Pig Smooth Muscles
Cingi, Munise İpek; Erol, K; Özdemir, M; Cingi, Cemal (Elsevier Science BV, 1990)… -
Effects of Ciprofloxacin on Chromosomes, and Hepatic and Renal Functions in Rats
Başaran, A; Erol, K; Başaran, N; Güneş, Hasan Veysi; Açıkalın, E; Timuralp, G; Tomatir, Ag (Karger, 1993)In the present study, ciprofloxacin, a fluoroquinolone antibiotic, was evaluated in vivo. The toxic effects of ciprofloxacin (20 and 200 mg/kg/day) on kidney and liver functions, and on chromosomes were investigated in ... -
Effects of Vasoactive Intestinal Polypeptide on Isolated Rat Urinary-Bladder Smooth-Muscle
The effect of vasoactive intestinal polypeptide (VIP) on the contractile activity of the urinary bladder was investigated in the rat. VIP caused a weak contraction and a small potentiation of carbachol- and acetylcholine-induced ... -
Gastroprotective Effect of Nitrendipine on Stress-Induced Gastric-Lesions in Rats
Ulak, G; Cingi, Munise İpek; Erol, K (Karger, 1991)The effects of nitrendipine on stress-induced acute gastric lesions were investigated in rats. Intraperitoneally injected nitrendipine (8, 16, or 32 mg/kg) given 30 min before stress, dose-dependently prevented gastric ... -
MgSO4 and lazaroid (U-83836E) partially protects glioma cells against glutamate toxicity in vitro
Kabadere, S; Öztopçu, P; Korkmaz, S; Erol, K; Uyar, R (Nencki Inst Experimental Biology, 2004)In this study, the possible effects Of MgSO4 and lazaroid (U-83836E) on glutamate toxicity on glial cells were investigated. C6 and human glioblastoma multiforme cells derived from two patients were grown in an incubator. ... -
Pharmacodynamic comparison of a nasal formulation of verapamil and intravenous and oral dosage forms
The nasal route has been shown to be effective for the administration of numerous drugs in order to improve drug bioavailability. A nasal gel of verapamil hydrochloride was formulated and evaluated pharmacodynamically in ... -
Reduction of Methotrexate Nephrotoxicity With Verapamil in Rats
Erol, K; Gürer, F; Bayçu, Cengiz; Cingi, Mi; Erol, A (Elsevier Science BV, 1990)… -
Studies on Some 10-[2-(N,N-Disubstituted Thiocarbamoylthio)Acetyl]Phenothiazine Derivatives
Palaska, E; Sarac, S; Şafak, C; Erdoğan, H; Erol, K; Alpan, Rs (Ecv-Editio Cantor Verlag Medizin Naturwissenschaften, 1992)Nineteen 10-[2-(NN-disubstituted thiocarbamolythio) acetyl]phenothiazine derivatives have been synthesized by the reaction of 10-chloroacetylphenothiazine with potassium salt of N,N-disubstituted dithiocarbamic acid ... -
Synthesis and Anticholinergic Activity of Some New N,N-Disubstituted Carbamodithioic Acid 2-Oxo-2-(Diphenylamino) Ethyl-Esters
Özkanli, F; Dalkara, S; Çalış, U; Erol, K; Özdemir, M (Soc Chimica Italiana, 1993)The synthesis of new N,N-disubstituted carbamodithioic acid 2-oxo-2-(diphenylamino) ethyl esters is reported. The structures of these compounds are supported by their UV, IR and H-1-NMR spectra, as well as by elemental ... -
Synthesis and Pharmacology of Some New Carbamodithioic Acid-Esters
Şafak, C; Erdoğan, H; Yeşilada, A; Erol, K; Cimgi, I (Georg Thieme Verlag Kg, 1992)In this study 13 new dithiocarbamates were prepared by reacting 3-methyl-6-chloroacetyl-benzoxazolinone with potassium N,N-disubstituted dithiocarbamate derivatives. The structures of the compounds were confirmed by UV, ... -
Synthesis and preliminary evaluation of new 5-pyrazolinone derivatives as analgesic agents
Gürsoy, A; Demirayak, Şeref; Capan, G; Erol, K; Vural, K (Editions Scientifiques Medicales Elsevier, 2000)New 4-(aroyloxyalkanoyl)-2,3-dimethyl-1-phenyl-3-pyrazolin-5-ones (5) were cyclized to 4-(2-aryl-5-unsubstituted/substituted oxazol-4-yl)-2,3-dimethyl-1-phenyl-3-pyrazolin-5-ones (6) employing the Davidson procedure. ... -
Synthesis of some triazolyl-antipyrine derivatives and investigation of analgesic activity
Turan, Gülhan; Sivaci, M; Kılıç, FS; Erol, K (Elsevier France-Editions Scientifiques Medicales Elsevier, 2001)The synthesis of some triazolyl-antipyrine derivatives starting from 4-chloroacetamidoantipyrine and 3-(aryloxyalkyl)-4-ethyl/phenyl-5-mercapto-1,2,4-triazoles is described. The chemical structures of the compounds were ...
